TargetMol

Brensocatib

Product Code:
 
TAR-TQ0038
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TQ0038-1mg1mg£124.00
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TAR-TQ0038-5mg5mg£201.00
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TAR-TQ0038-1mL1 mL * 10 mM (in DMSO)£213.00
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TAR-TQ0038-10mg10mg£302.00
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TAR-TQ0038-25mg25mg£460.00
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TAR-TQ0038-50mg50mg£627.00
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This product comes from: United States.
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Further Information

Bioactivity:
AZD7986 is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).
CAS:
1802148-05-5
Formula:
C23H24N4O4
Molecular Weight:
420.469
Pathway:
Proteases/Proteasome; Ubiquitination
Purity:
0.9905
SMILES:
Cn1c2cc(ccc2oc1=O)-c1ccc(C[C@H](NC(=O)[C@@H]2CNCCCO2)C#N)cc1
Target:
Proteasome

References

Doyle K, et al. Discovery of Second Generation Reversible Covalent DPP1 Inhibitors Leading to an Oxazepane Amidoacetonitrile Based Clinical Candidate (AZD7986). J Med Chem. 2016 Oct 27;59(20):9457-9472.