TargetMol

LY2795050

Product Code:
 
TAR-TQ0091
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TQ0091-1mg1mg£135.00
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TAR-TQ0091-2mg2mg£164.00
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TAR-TQ0091-5mg5mg£229.00
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TAR-TQ0091-1mL1 mL * 10 mM (in DMSO)£244.00
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TAR-TQ0091-10mg10mg£325.00
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TAR-TQ0091-25mg25mg£490.00
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TAR-TQ0091-50mg50mg£670.00
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This product comes from: United States.
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Further Information

Bioactivity:
LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).
CAS:
1346133-08-1
Formula:
C23H22ClN3O2
Molecular Weight:
407.9
Pathway:
Endocrinology/Hormones; GPCR/G Protein; Neuroscience
Purity:
0.9777
SMILES:
NC(=O)c1ccc(Oc2ccc(CN3CCCC3c3cccnc3)cc2)c(Cl)c1
Target:
Opioid Receptor

References

Mitch, Charles H.; Quimby, Steven J.; Diaz, Nuria; et al. Discovery of Aminobenzyloxyarylamides as ? Opioid Receptor Selective Antagonists: Application to Preclinical Development of a ? Opioid Receptor Antagonist Receptor Occupancy Tracer. Journal of Medicinal Chemistry (2011), 54(23), 8000-8012. Zheng MQ, Nabulsi N, Kim SJ, Synthesis and evaluation of 11C-LY2795050 as a ?-opioid receptor antagonist radiotracer for PET imaging. J Nucl Med. 2013 Mar;54(3):455-63.