TargetMol

ETP-46321

Product Code:
 
TAR-TQ0229
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TQ0229-1mg1mg£148.00
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TAR-TQ0229-5mg5mg£282.00
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TAR-TQ0229-1mL1 mL * 10 mM (in DMSO)£302.00
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TAR-TQ0229-10mg10mg£389.00
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TAR-TQ0229-25mg25mg£603.00
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TAR-TQ0229-50mg50mg£830.00
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TAR-TQ0229-100mg100mg£1,099.00
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TAR-TQ0229-500mg500mg£2,135.00
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This product comes from: United States.
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Further Information

Bioactivity:
ETP-46321 is an effective and orally bioavailable PI3Kα/PI3Kδ inhibitor (Ki: 2.3/14.2 nM).
CAS:
1252594-99-2
Formula:
C20H27N9O3S
Molecular Weight:
473.56
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.9947
SMILES:
CS(=O)(=O)N1CCN(Cc2cn3cc(nc(N4CCOCC4)c3n2)-c2cnc(N)nc2)CC1
Target:
PI3K

References

Mart?nez Gonz?lez S, et al. Identification of ETP-46321, a potent and orally bioavailable PI3K ?, ? inhibitor. Bioorg Med Chem Lett. 2012 May 15;22(10):3460-6.