TargetMol

BIBF 1202

Product Code:
 
TAR-TQ0321
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
BIBF 1202 is a VEGFR2 kinase inhibitor (IC50 = 62 nM).
CAS:
894783-71-2
Formula:
C30H31N5O4
Molecular Weight:
525.609
Pathway:
Angiogenesis; Tyrosine Kinase/Adaptors
Purity:
0.98
SMILES:
CN(C(=O)CN1CCN(C)CC1)c1ccc(NC(=C2/C(=O)Nc3cc(ccc23)C(O)=O)c2ccccc2)cc1
Target:
VEGFR

References

Hilberg F, et al. BIBF 1120: triple angiokinase inhibitor with sustained receptor blockade and good antitumorefficacy. Cancer Res. 2008 Jun 15;68(12):4774-82. Stopfer P, et al. Pharmacokinetics and metabolism of BIBF 1120 after oral dosing to healthy male volunteers. Xenobiotica. 2011 Apr;41(4):297-311.