TargetMol

Pimethixene

Product Code:
 
TAR-T12489
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12489-1mg1mg£99.00
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TAR-T12489-2mg2mg£109.00
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TAR-T12489-5mg5mg£128.00
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TAR-T12489-1mL1 mL * 10 mM (in DMSO)£136.00
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TAR-T12489-10mg10mg£152.00
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TAR-T12489-25mg25mg£215.00
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TAR-T12489-50mg50mg£285.00
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TAR-T12489-100mg100mg£389.00
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TAR-T12489-200mg200mg£547.00
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TAR-T12489-500mg500mg£833.00
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This product comes from: United States.
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Further Information

Bioactivity:
Pimethixene is a highly potent 5-HT1A, 5-HT2A, 5-HT2B, 5-HT2C, histamine H1, dopamine D2 and D4.4 as well as muscarinic M1 and M2 receptors antagonist(pKis of 7.63, 10.22, 10.44, 8.42, 10.14, 8.19, 7.54, 8.61 and 9.38, respectively).
CAS:
314-03-4
Formula:
C19H19NS
Molecular Weight:
293.43
Pathway:
GPCR/G Protein; Immunology/Inflammation; Neuroscience
Purity:
0.991
SMILES:
CN1CCC(CC1)=C1c2ccccc2Sc2ccccc12
Target:
Dopamine Receptor; 5-HT Receptor; AChR; Histamine Receptor

References

1. Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80.