TargetMol

Seltorexant

Product Code:
 
TAR-T12877L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
❮❯

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CodeSizePrice
TAR-T12877L-1mg1mg£101.00
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TAR-T12877L-2mg2mg£114.00
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TAR-T12877L-5mg5mg£142.00
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TAR-T12877L-1mL1 mL * 10 mM (in DMSO)£148.00
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TAR-T12877L-10mg10mg£177.00
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TAR-T12877L-25mg25mg£233.00
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TAR-T12877L-50mg50mg£362.00
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TAR-T12877L-100mg100mg£503.00
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TAR-T12877L-500mg500mg£1,018.00
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Further Information

Bioactivity:
Seltorexant crosses the blood-brain barrier and quickly occupies OX2R binding sites in the rat brain. Seltorexant is a high-affinity and selective orexin-2 receptor antagonist (pKi: 8.0 and 8.1 for human and rat OX2R).
CAS:
1293281-49-8
Formula:
C21H22FN7O
Molecular Weight:
407.453
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9979
SMILES:
Cc1cc(C)nc(n1)N1CC2CN(CC2C1)C(=O)c1c(F)cccc1-n1nccn1
Target:
OX Receptor

References

1. Bonaventure P, et al. Characterization of JNJ-42847922, a Selective Orexin-2 Receptor Antagonist, as a Clinical Candidate for the Treatment of Insomnia. J Pharmacol Exp Ther. 2015 Sep;354(3):471-82.