TargetMol

Fezagepras

Product Code:
 
TAR-T12883
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T12883-100mg100mgEnquire
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Quantity:
TAR-T12883-1mg1mg£109.00
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TAR-T12883-2mg2mg£125.00
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TAR-T12883-1mL1 mL * 10 mM (in DMSO)£146.00
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TAR-T12883-5mg5mg£148.00
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TAR-T12883-10mg10mg£185.00
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Quantity:
TAR-T12883-25mg25mg£278.00
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Quantity:
TAR-T12883-50mg50mg£367.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Setogepram is an orally active GPR40 agonist and is an antagonist or inverse agonist of GPR84 with anti-inflammatory, anti-fibrotic, and anti-proliferative actions.
CAS:
1002101-19-0
Formula:
C13H18O2
Molecular Weight:
206.285
Pathway:
Endocrinology/Hormones; GPCR/G Protein
Purity:
0.9938
SMILES:
CCCCCc1cccc(CC(O)=O)c1
Target:
GPR

References

1. Li Y, et al. Fatty acid receptor modulator PBI-4050 inhibits kidney fibrosis and improves glycemic control. JCI Insight. 2018 May 17;3(10). pii: 120365. 2. Grouix B, et al. PBI-4050 Reduces Stellate Cell Activation and Liver Fibrosis through Modulation of Intracellular ATP Levels and the Liver Kinase B1/AMP-Activated Protein Kinase/Mammalian Target of Rapamycin Pathway. J Pharmacol Exp Ther. 2018 Oct;367(1):71-81.