TargetMol

TAK-071

Product Code:
 
TAR-T13066
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T13066-1mg1mg£101.00
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TAR-T13066-2mg2mg£114.00
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TAR-T13066-5mg5mg£141.00
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TAR-T13066-1mL1 mL * 10 mM (in DMSO)£157.00
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TAR-T13066-10mg10mg£182.00
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TAR-T13066-25mg25mg£267.00
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TAR-T13066-50mg50mg£386.00
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TAR-T13066-100mg100mg£540.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).
CAS:
1820812-16-5
Formula:
C24H24FN3O3
Molecular Weight:
421.472
Pathway:
Neuroscience
Purity:
0.9847
SMILES:
Cc1c(F)c2CN([C@H]3COCC[C@@H]3O)C(=O)c2cc1Cc1ccc(cc1)-n1cccn1
Target:
AChR

References

1. Sako Y, et al. TAK-071, a novel M1 positive allosteric modulator with low cooperativity, improves cognitive function in rodents with few cholinergic side effects. Neuropsychopharmacology. 2018 Aug doi: 10.1038/s41386-018-0168-8.