TargetMol

VU6005649

Product Code:
 
TAR-T13321
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13321-1mg1mg£95.00
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TAR-T13321-2mg2mg£106.00
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TAR-T13321-5mg5mg£128.00
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TAR-T13321-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T13321-10mg10mg£168.00
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TAR-T13321-25mg25mg£282.00
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TAR-T13321-50mg50mg£484.00
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TAR-T13321-100mg100mg£695.00
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Quantity:
TAR-T13321-500mg500mg£1,348.00
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This product comes from: United States.
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Further Information

Bioactivity:
VU6005649 is an agonist of CNS penetrant mGlu7/8 receptor (EC50s: 0.65 μM and 2.6 μM for mGlu7 receptor and mGlu8 receptor, respectively).
CAS:
2137047-43-7
Formula:
C16H12F5N3O
Molecular Weight:
357.284
Pathway:
Neuroscience
Purity:
0.98
SMILES:
COc1ccc(-c2c(C)nn3c(cc(C)nc23)C(F)(F)F)c(F)c1F
Target:
GluR

References

1. Abe M, et al. Discovery of VU6005649, a CNS Penetrant mGlu7/8 Receptor PAM Derived from a Series of Pyrazolo[1,5-a]pyrimidines. ACS Med Chem Lett. 2017 Sep 1;8(10):1110-1115.