TargetMol

VU6012962

Product Code:
 
TAR-T13323
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T13323-1mg1mg£95.00
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TAR-T13323-2mg2mg£106.00
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TAR-T13323-5mg5mg£128.00
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TAR-T13323-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T13323-10mg10mg£173.00
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TAR-T13323-25mg25mg£270.00
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TAR-T13323-50mg50mg£430.00
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TAR-T13323-100mg100mg£599.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
VU6012962 is an orally bioavailable negative allosteric modulator of CNS-penetrant metabotropic glutamate receptor 7(mGlu7; IC50: 347 nM).
CAS:
2313526-86-0
Formula:
C21H19F3N4O4
Molecular Weight:
448.4
Pathway:
Neuroscience
Purity:
0.98
SMILES:
COC1=C(C=CC(=C1)C(=O)NC2=C(C=CC(=C2)OC(F)(F)F)N3C=NC=N3)OCC4CC4
Target:
GluR

References

1. Reed CW, et al. Discovery of an orally bioavailable and Central Nervous System (CNS) penetrant mGlu7 NegativeAllosteric Modulator (NAM) in vivo tool compound: N-(2-(1H-1,2,4-triazol-1-yl)-5-(trifluoromethoxy)phenyl)-4-(cyclopropylmethoxy)-3-methoxybenzamide (VU6012962). J Med Chem. 2019 Jan 4.