TargetMol

CaMKII-IN-1

Product Code:
 
TAR-T14860
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T14860-1mg1mg£109.00
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TAR-T14860-2mg2mg£125.00
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TAR-T14860-5mg5mg£168.00
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TAR-T14860-1mL1 mL * 10 mM (in DMSO)£189.00
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TAR-T14860-10mg10mg£213.00
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TAR-T14860-25mg25mg£369.00
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TAR-T14860-50mg50mg£535.00
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TAR-T14860-100mg100mg£740.00
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Further Information

Bioactivity:
CaMKII-IN-1 is a potent and highly selective inhibitor of CaMKII (IC50 = 63 nM). CaMKII-IN-1 exhibited more than 100-fold higher selectivity for CaMKII over CaMKIV, MLCK, p38a, Akt1, and PKC.
CAS:
1208123-85-6
Formula:
C29H30ClN5O2S
Molecular Weight:
548.1
Pathway:
Autophagy; Neuroscience
Purity:
0.9835
SMILES:
Cc1c(Cl)cccc1S(=O)(=O)Nc1nc(NCCc2ccccc2)nc2CCN(Cc3ccccc3)Cc12
Target:
CaMK; Autophagy

References

1. Asano S, et al. 5,6,7,8-Tetrahydropyrido[4,3-d]pyrimidines as novel class of potent and highly selective CaMKII inhibitors. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6696-8.