TargetMol

PROTAC ERR α ligand 1

Product Code:
 
TAR-T15191
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15191-1mg1mg£106.00
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TAR-T15191-2mg2mg£121.00
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TAR-T15191-5mg5mg£148.00
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TAR-T15191-1mL1 mL * 10 mM (in DMSO)£164.00
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TAR-T15191-10mg10mg£189.00
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TAR-T15191-25mg25mg£282.00
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TAR-T15191-50mg50mg£414.00
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TAR-T15191-100mg100mg£584.00
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TAR-T15191-500mg500mg£1,171.00
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Further Information

Bioactivity:
PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
CAS:
1264754-13-3
Formula:
C19H11F3N2O4S
Molecular Weight:
420.36
Pathway:
Endocrinology/Hormones
Purity:
0.9945
SMILES:
N#CC1=CC=C(OC2=CC=C(/C=C(SC(N3)=O)/C3=O)C=C2OC)C(C(F)(F)F)=C1
Target:
Estrogen Receptor/ERR; Estrogen/progestogen Receptor

References

1. Patch RJ, et al. Identification of diaryl ether-based ligands for estrogen-related receptor ? as potential antidiabetic agents. J Med Chem. 2011 Feb 10;54(3):788-808.