TargetMol

GSK2837808A

Product Code:
 
TAR-T15435
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15435-1mg1mg£103.00
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TAR-T15435-5mg5mg£170.00
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TAR-T15435-1mL1 mL * 10 mM (in DMSO)£213.00
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TAR-T15435-10mg10mg£229.00
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TAR-T15435-25mg25mg£438.00
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TAR-T15435-50mg50mg£457.00
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Quantity:
TAR-T15435-100mg100mg£631.00
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This product comes from: United States.
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Further Information

Bioactivity:
GSK2837808A is a potent and selective inhibitor of lactate dehydrogenase A (LDHA) (IC50s: 1.9 and 14 nM for LDHA and LDHB, respectively).
CAS:
1445879-21-9
Formula:
C31H25F2N5O7S
Molecular Weight:
649.63
Pathway:
Metabolism
Purity:
0.9978
SMILES:
COc1ncc(-c2ccc3c(Nc4cc(Oc5cc(F)cc(F)c5)cc(c4)C(O)=O)c(cnc3c2)S(=O)(=O)NC2CC2)c(OC)n1
Target:
Dehydrogenase

References

1. Billiard J, et al. Quinoline 3-sulfonamides inhibit lactate dehydrogenase A and reverse aerobic glycolysis in cancer cells. Cancer Metab. 2013 Sep 6;1(1):19.