TargetMol

KH7

Product Code:
 
TAR-T15658
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15658-50mg50mgEnquire
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TAR-T15658-1mg1mg£100.00
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TAR-T15658-2mg2mg£111.00
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TAR-T15658-5mg5mg£136.00
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TAR-T15658-1mL1 mL * 10 mM (in DMSO)£144.00
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TAR-T15658-10mg10mg£177.00
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TAR-T15658-25mg25mg£283.00
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Further Information

Bioactivity:
KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific. It has IC50s of 3-10 μM toward both recombinant purified human sACt protein and heterologously expressed sACt in cellular assays. KH7 is also a cAMP inhibitor.
CAS:
330676-02-3
Formula:
C17H15BrN4O2S
Molecular Weight:
419.3
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9956
SMILES:
CC(Sc1nc2ccccc2[nH]1)C(=O)NN=Cc1cc(Br)ccc1O
Target:
cAMP; AChR

References

1. Hess KC, et al. The "soluble" adenylyl cyclase in sperm mediates multiple signaling events required for fertilization. Dev Cell. 2005 Aug;9(2):249-59. 2. Han J, et al. Maresin Conjugates in Tissue Regeneration 1 improves alveolar fluid clearance by up-regulating alveolar ENaC, Na, K-ATPase in lipopolysaccharide-induced acute lung injury. 4.658J Cell Mol Med. 2020 Mar 11.