TargetMol

Laropiprant

Product Code:
 
TAR-T15712
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T15712-1mg1mg£114.00
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TAR-T15712-2mg2mg£133.00
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TAR-T15712-5mg5mg£177.00
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TAR-T15712-1mL1 mL * 10 mM (in DMSO)£187.00
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TAR-T15712-10mg10mg£225.00
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TAR-T15712-25mg25mg£380.00
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TAR-T15712-50mg50mg£546.00
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TAR-T15712-100mg100mg£749.00
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TAR-T15712-500mg500mg£1,428.00
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Further Information

Bioactivity:
Laropiprant is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such as and DP/DP1 receptor(Ki = 0.57 nM) and TP Receptor(Ki = 2.95 nM).
CAS:
571170-77-9
Formula:
C21H19ClFNO4S
Molecular Weight:
435.9
Pathway:
Immunology/Inflammation; GPCR/G Protein
Purity:
0.98
SMILES:
O=S(C1=CC(F)=CC2=C1N(C3=C2CC[C@@H]3CC(O)=O)CC4=CC=C(Cl)C=C4)(C)=O
Target:
Prostaglandin Receptor

References

1. Sturino CF, et al. Discovery of a potent and selective prostaglandin D2 receptor antagonist, [(3R)-4-(4-chloro-benzyl)-7-fluoro-5-(methylsulfonyl)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl]-acetic acid (MK-0524). J Med Chem. 2007 Feb 22;50(4):794-806. 2. Philipose S, et al. Laropiprant Attenuates EP3 and TP Prostanoid Receptor-Mediated Thrombus Formation. PLoS One. 2012;7(8):e40222.