TargetMol

(S,R,S)-AHPC-PEG3-NH2 hydrochloride

Product Code:
 
TAR-T17922
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T17922-5mg5mg£102.00
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Quantity:
TAR-T17922-10mg10mg£122.00
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Quantity:
TAR-T17922-25mg25mg£173.00
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TAR-T17922-50mg50mg£262.00
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Quantity:
TAR-T17922-100mg100mg£434.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
(S,R,S)-AHPC-PEG3-NH2 hydrochloride is an E3 ligase ligand-linker conjugate incorporating the (S,R,S)-AHPC-based VHL ligand and 3-unit PEG linker.
CAS:
2097971-11-2
Formula:
C30H46ClN5O7S
Molecular Weight:
656.23
Pathway:
Others|PROTAC
Purity:
0.9758
SMILES:
NCCOCCOCCOCC(N[C@@H](C(C)(C)C)C(N1[C@@H](C[C@H](C1)O)C(NCC2=CC=C(C3=C(N=CS3)C)C=C2)=O)=O)=O.Cl
Target:
Others|E3 Ligase Ligand-Linker Conjugate

References

1. Chan KH, et al. Impact of Target Warhead and Linkage Vector on Inducing Protein Degradation: Comparison of Bromodomain and Extra-Terminal (BET) Degraders Derived from Triazolodiazepine (JQ1) and Tetrahydroquinoline (I-BET726) BET Inhibitor Scaffolds. J Med Chem. 2018 Jan 25;61(2):504-513.