TargetMol

BX-912

Product Code:
 
TAR-T1837
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T1837-1mg1mg£109.00
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TAR-T1837-2mg2mg£125.00
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TAR-T1837-5mg5mg£136.00
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TAR-T1837-1mL1 mL * 10 mM (in DMSO)£139.00
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TAR-T1837-10mg10mg£189.00
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TAR-T1837-25mg25mg£322.00
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TAR-T1837-50mg50mg£490.00
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TAR-T1837-100mg100mg£635.00
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This product comes from: United States.
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Further Information

Bioactivity:
BX-912 is a specific inhibitor of 3-Phosphoinositide-dependent Kinase-1 (PDK1, IC50: 12 nM). The selectivity of BX-912 is more 10 fold than C-Kit, EGFR, PKA, PKC etc.
CAS:
702674-56-4
Formula:
C20H23BrN8O
Molecular Weight:
471.363
Pathway:
Angiogenesis; Cell Cycle/Checkpoint; PI3K/Akt/mTOR signaling; Tyrosine Kinase/Adaptors; Apoptosis
Purity:
0.9934
SMILES:
Brc1cnc(Nc2cccc(NC(=O)N3CCCC3)c2)nc1NCCc1c[nH]cn1
Target:
Apoptosis; VEGFR; PKA; Chk; CDK; PDK

References

1. Feldman RI, et al. J Biol Chem. 2005, 280(20), 19867-19874.