TargetMol

Fimepinostat

Product Code:
 
TAR-T2078
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2078-2mg2mg£102.00
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TAR-T2078-5mg5mg£122.00
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TAR-T2078-1mL1 mL * 10 mM (in DMSO)£128.00
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TAR-T2078-10mg10mg£149.00
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TAR-T2078-25mg25mg£219.00
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TAR-T2078-50mg50mg£334.00
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TAR-T2078-100mg100mg£503.00
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TAR-T2078-500mg500mg£994.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
CUDC-907 is an orally bioavailable inhibitor of both phosphoinositide 3-kinase (PI3K) class I and pan-histone deacetylase (HDAC) enzymes, with potential antineoplastic activity. Upon oral administration, CUDC-907 inhibits the activity of both PI3K class I isoforms and HDAC, thereby preventing the activation of the PI3K-AKT-mTOR signal transduction pathway that is often overactivated in many cancer cell types.
CAS:
1339928-25-4
Formula:
C23H24N8O4S
Molecular Weight:
508.56
Pathway:
Apoptosis; PI3K/Akt/mTOR signaling; Chromatin/Epigenetic; DNA Damage/DNA Repair
Purity:
0.9966
SMILES:
COc1ccc(cn1)-c1nc(N2CCOCC2)c2sc(CN(C)c3ncc(cn3)C(=O)NO)cc2n1
Target:
Apoptosis; PI3K; HDAC

References

1. Qian C, et al. Cancer network disruption by a single molecule inhibitor targeting both histone deacetylase activity and phosphatidylinositol 3-kinase signaling. Clin Cancer Res. 2012 Aug 1;18(15):4104-13.