TargetMol

1-NM-PP1

Product Code:
 
TAR-T2153
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2153-1mg1mg£105.00
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TAR-T2153-2mg2mg£119.00
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TAR-T2153-5mg5mg£136.00
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TAR-T2153-1mL1 mL * 10 mM (in DMSO)£140.00
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TAR-T2153-10mg10mg£185.00
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TAR-T2153-25mg25mg£313.00
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Quantity:
TAR-T2153-50mg50mg£520.00
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Quantity:
TAR-T2153-100mg100mg£667.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
1 nM-PP1 is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.
CAS:
221244-14-0
Formula:
C20H21N5
Molecular Weight:
331.423
Pathway:
Metabolism; Cell Cycle/Checkpoint; Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.992
SMILES:
CC(C)(C)n1nc(Cc2cccc3ccccc23)c2c(N)ncnc12
Target:
Serine/threonin kinase; CDK; Src

References

1. Larochelle S, et al. Requirements for Cdk7 in the assembly of Cdk1/cyclin B and activation of Cdk2 revealed by chemical genetics in human cells. Mol Cell. 2007 Mar 23;25(6):839-50.