TargetMol

AS1269574

Product Code:
 
TAR-T21623
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T21623-2mg2mg£103.00
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TAR-T21623-5mg5mg£122.00
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TAR-T21623-1mL1 mL * 10 mM (in DMSO)£135.00
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TAR-T21623-10mg10mg£158.00
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TAR-T21623-25mg25mg£237.00
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TAR-T21623-50mg50mg£334.00
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TAR-T21623-100mg100mg£464.00
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TAR-T21623-500mg500mg£946.00
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Further Information

Bioactivity:
AS 1269574 is a potent, orally available GPR119 agonist. AS1269574 has the potential for the research of type 2 diabetes.
CAS:
330981-72-1
Formula:
C13H14BrN3O
Molecular Weight:
308.18
Pathway:
GPCR/G Protein; Membrane transporter/Ion channel; Endocrinology/Hormones
Purity:
0.9998
SMILES:
CC1=CC(=NC(=N1)C2=CC=C(C=C2)Br)NCCO
Target:
GPR; TRP/TRPV Channel

References

1. Yoshida S, et al. Identification of a novel GPR119 agonist, AS1269574, with in vitro and in vivo glucose-stimulated insulin secretion. Biochem Biophys Res Commun. 2010;400(3):437-441. 2. Chepurny OG, et al. GPR119 Agonist AS1269574 Activates TRPA1 Cation Channels to Stimulate GLP-1 Secretion. Mol Endocrinol. 2016;30(6):614-629.