TargetMol

PD184161

Product Code:
 
TAR-T21635
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T21635-1mg1mg£96.00
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TAR-T21635-2mg2mg£106.00
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TAR-T21635-5mg5mg£128.00
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TAR-T21635-10mg10mg£173.00
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TAR-T21635-25mg25mg£301.00
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TAR-T21635-50mg50mg£454.00
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Quantity:
TAR-T21635-100mg100mg£623.00
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TAR-T21635-200mg200mg£863.00
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Quantity:
TAR-T21635-500mg500mg£1,259.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PD184161 is a novel, orally-active MEK inhibitor. PD184161 inhibited MEK activity (IC50 = 10-100 nM) in a time- and concentration-dependent manner[1].
CAS:
212631-67-9
Formula:
C17H13BrClF2IN2O2
Molecular Weight:
557.56
Pathway:
MAPK
Purity:
0.9909
SMILES:
Fc1c(F)c(Nc2ccc(I)cc2Cl)c(cc1Br)C(=O)NOCC1CC1
Target:
MEK

References

1. Klein, P. J.,Schmidt, C.M.,Wiesenauer, C.A., et al. The effects of a novel MEK inhibitor PD184161 on MEK-ERK signaling and growth in human liver cancer. Neoplasia 8(1), 1-8 (2006).