TargetMol

ARC 239 dihydrochloride

Product Code:
 
TAR-T22033
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T22033-1mg1mg£97.00
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TAR-T22033-5mg5mg£132.00
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TAR-T22033-1mL1 mL * 10 mM (in DMSO)£148.00
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TAR-T22033-10mg10mg£177.00
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TAR-T22033-25mg25mg£298.00
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TAR-T22033-50mg50mg£436.00
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TAR-T22033-100mg100mg£598.00
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This product comes from: United States.
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Further Information

Bioactivity:
ARC 239 dihydrochloride is a selective α2B adrenoceptor antagonist (pKD values are 8.8, 6.7 and 6.4 at α2B, α2A, and α2D receptors respectively).
CAS:
55974-42-0
Formula:
C24H31Cl2N3O3
Molecular Weight:
480.43
Pathway:
Neuroscience
Purity:
0.98
SMILES:
O=C(N1CCN2CCN(C(C=CC=C3)=C3OC)CC2)C4=CC=CC=C4C(C)(C)C1=O.Cl.Cl
Target:
Norepinephrine

References

1. Suzana Assad Kahn, et al. The anti-hypertensive drug prazosin inhibits glioblastoma growth via the PKC?-dependent inhibition of the AKT pathway. EMBO Mol Med. 2016 May 2;8(5):511-26.