TargetMol

HA-155

Product Code:
 
TAR-T22086
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T22086-1mg1mg£107.00
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TAR-T22086-2mg2mg£120.00
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TAR-T22086-5mg5mg£177.00
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TAR-T22086-10mg10mg£261.00
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TAR-T22086-25mg25mg£527.00
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TAR-T22086-50mg50mg£645.00
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Quantity:
TAR-T22086-100mg100mg£772.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
HA155 is a boronic acid-based compound, inhibiting ATX with IC50 of 5.7 nM by selectively binding to its catalytic threonine.
CAS:
1229652-22-5
Formula:
C24H19BFNO5S
Molecular Weight:
463.29
Pathway:
Metabolism
Purity:
0.9892
SMILES:
B(C1=CC=C(C=C1)COC2=CC=C(C=C2)/C=C3/C(=O)N(C(=O)S3)CC4=CC=C(C=C4)F)(O)O
Target:
PDE

References

1. Albers H M H G , Hendrickx L J D , Van Tol R J P , et al. Structure-Based Design of Novel Boronic Acid-Based Inhibitors of Autotaxin[J]. Journal of Medicinal Chemistry, 2011, 54(13):4619-26.