TargetMol

DGY-06-116

Product Code:
 
TAR-T22306
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T22306-1mg1mg£103.00
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TAR-T22306-2mg2mg£118.00
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TAR-T22306-5mg5mg£148.00
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TAR-T22306-1mL1 mL * 10 mM (in DMSO)£156.00
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TAR-T22306-10mg10mg£201.00
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TAR-T22306-25mg25mg£329.00
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TAR-T22306-50mg50mg£470.00
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TAR-T22306-100mg100mg£670.00
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Further Information

Bioactivity:
DGY-06-116 is an selective and irreversible covalent inhibitor of Src and FGFR1 with IC50 value of 3nM and 8340 nM, respectively.
CAS:
T22306
Formula:
C32H33ClN8O2
Molecular Weight:
597.11
Pathway:
Angiogenesis; Tyrosine Kinase/Adaptors
Purity:
0.996
SMILES:
CN1CCN(CC1)c1ccc(Nc2ncc(C(=O)Nc3c(C)cccc3Cl)c(Nc3ccccc3NC(=O)C=C)n2)cc1
Target:
FGFR; Src

References

1. Gurbani D , Du G , Henning N J , et al. Structure and Characterization of a Covalent Inhibitor of Src Kinase[J]. Frontiers in Molecular Bioences, 2020, 7:81.