TargetMol

CID755673

Product Code:
 
TAR-T2458
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T2458-2mg2mg£99.00
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TAR-T2458-5mg5mg£113.00
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TAR-T2458-1mL1 mL * 10 mM (in DMSO)£116.00
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TAR-T2458-10mg10mg£132.00
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TAR-T2458-25mg25mg£173.00
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TAR-T2458-50mg50mg£237.00
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Quantity:
TAR-T2458-100mg100mg£367.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective PKD1 inhibition when compared with PLK1, AKT, CAMKIIα, CAK, and PKC isoforms.
CAS:
521937-07-5
Formula:
C12H11NO3
Molecular Weight:
217.224
Pathway:
Cell Cycle/Checkpoint; Metabolism
Purity:
0.9984
SMILES:
Oc1ccc2oc3c(CCCNC3=O)c2c1
Target:
Serine/threonin kinase

References

1. Sharlow ER, et al. J Biol Chem. 2008, 283(48), 33516-33526. 2. Yuan J, et al. Front Physiol. 2012, 3, 60. 3. Scheiter M, et al. Front Immunol. 2013, 4, 66.