TargetMol

JNJ-42165279

Product Code:
 
TAR-T3215
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T3215-1mg1mg£107.00
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TAR-T3215-2mg2mg£122.00
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TAR-T3215-5mg5mg£152.00
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TAR-T3215-1mL1 mL * 10 mM (in DMSO)£165.00
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TAR-T3215-10mg10mg£191.00
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TAR-T3215-25mg25mg£302.00
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Quantity:
TAR-T3215-50mg50mg£417.00
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TAR-T3215-100mg100mg£581.00
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Quantity:
TAR-T3215-200mg200mg£792.00
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Quantity:
TAR-T3215-500mg500mg£1,155.00
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Further Information

Bioactivity:
JNJ-42165279 covalently inactivates the FAAH enzyme but is highly selective with regard to other enzymes, ion channels, transporters, and receptors. JNJ-42165279 (10 μM) exhibits high selectivity against a panel of 50 receptors, enzymes, transporters, and ion-channels, at which concentration it does not produce >50% inhibition of binding to any of the targets. Fortunately, JNJ-42165279 (10 μM) also does not inhibit CYPs (1A2, 2C8, 2C9, 2C19, 2D6, 3A4) or hERG.
CAS:
1346528-50-4
Formula:
C18H17ClF2N4O3
Molecular Weight:
410.81
Pathway:
Autophagy; Metabolism; Neuroscience
Purity:
0.9991
SMILES:
FC1(F)Oc2ccc(CN3CCN(CC3)C(=O)Nc3cnccc3Cl)cc2O1
Target:
FAAH; Autophagy

References

1. Keith JM, et al. ACS Med Chem Lett. 2015 Nov 2;6(12):1204-8.