TargetMol

PEAQX

Product Code:
 
TAR-T4171
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4171-1mg1mg£107.00
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TAR-T4171-2mg2mg£122.00
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TAR-T4171-5mg5mg£164.00
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TAR-T4171-1mL1 mL * 10 mM (in DMSO)£205.00
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TAR-T4171-10mg10mg£240.00
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TAR-T4171-25mg25mg£376.00
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TAR-T4171-50mg50mg£545.00
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TAR-T4171-100mg100mg£748.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
PEAQX(NVP-AAM 077) is an effective and orally available NMDA antagonist. It can inhibit human NMDA receptors for 1A/2A(IC50: 270 nM), rather than 1A/2B(29, 600 nM).
CAS:
459836-30-7
Formula:
C17H17BrN3O5P
Molecular Weight:
454.217
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.98
SMILES:
C[C@H](NC(c1cccc2[nH]c(=O)c(=O)[nH]c12)P(O)(O)=O)c1ccc(Br)cc1
Target:
NMDAR; iGluR

References

Anastasio NC, et al. Differential role of N-methyl-D-aspartate receptor subunits 2A and 2B in mediating phencyclidine-induced perinatal neuronal apoptosis and behavioral deficits. Neuroscience. 2009 Nov 10;163(4):1181-91. Auberson YP, et al. 5-Phosphonomethylquinoxalinediones as competitive NMDA receptor antagonists with a preference for the human 1A/2A, rather than 1A/2B receptor composition. Bioorg Med Chem Lett. 2002 Apr 8;12(7):1099-102.