TargetMol

Betrixaban hydrochloride(330942-05-7(free base))

Product Code:
 
TAR-T4690
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T4690-1mg1mg£103.00
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TAR-T4690-2mg2mg£115.00
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TAR-T4690-5mg5mg£149.00
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TAR-T4690-1mL1 mL * 10 mM (in DMSO)£157.00
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TAR-T4690-10mg10mg£196.00
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TAR-T4690-25mg25mg£356.00
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TAR-T4690-50mg50mg£510.00
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TAR-T4690-100mg100mg£703.00
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This product comes from: United States.
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Further Information

Bioactivity:
Betrixaban is a potent, selective, and orally efficacious factor Xa (fXa) inhibitor (IC50: 1.5 nM).
CAS:
T4690
Formula:
C23H23Cl2N5O3
Molecular Weight:
488.36
Pathway:
Metabolism
Purity:
0.9954
SMILES:
Cl.COc1ccc(NC(=O)c2ccc(cc2)C(=N)N(C)C)c(c1)C(=O)Nc1ccc(Cl)cn1
Target:
Factor Xa

References

Zhang P, et al. Discovery of Betrixaban (PRT054021), N-(5-chloropyridin-2-yl)-2-(4-(N,N-dimethylcarbamimidoyl)benzamido)-5-methoxybenzamide, a highly potent, selective, and orally efficacious factor Xa inhibitor. Bioorg Med Chem Lett. 2009 Apr 15;19(8):2179-85. Lu G, et al. A specific antidote for reversal of anticoagulation by direct and indirect inhibitors of coagulation factor Xa. Nat Med. 2013 Apr;19(4):446-51.