TargetMol

WDR5-0103 hydrochloride[890190-22-4(free base)]

Product Code:
 
TAR-T5140
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T5140-1mg1mg£100.00
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Quantity:
TAR-T5140-2mg2mg£111.00
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TAR-T5140-5mg5mg£124.00
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TAR-T5140-10mg10mg£168.00
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TAR-T5140-25mg25mg£246.00
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TAR-T5140-50mg50mg£375.00
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Quantity:
TAR-T5140-100mg100mg£452.00
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Quantity:
TAR-T5140-200mg200mg£629.00
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Quantity:
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This product comes from: United States.
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Further Information

Bioactivity:
WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd: 450 nM).
CAS:
T5140
Formula:
C21H26ClN3O4
Molecular Weight:
419.9
Pathway:
JAK/STAT signaling; Angiogenesis; Chromatin/Epigenetic; Stem Cells
Purity:
0.9981
SMILES:
Cl.COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cccc(OC)c2)c1
Target:
JAK

References

Senisterra G, et al. Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5. Biochem J. 2013 Jan 1;449(1):151-159.