TargetMol

V-0219

Product Code:
 
TAR-T60047
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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Further Information

Bioactivity:
V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
CAS:
878453-71-5
Formula:
C20H25F3N4O2
Molecular Weight:
410.43
Pathway:
GPCR/G Protein
Purity:
1
SMILES:
FC(F)(F)C=1C=CC(=CC1)C2=NOC(=N2)CN3CCCC(C3)CN4CCOCC4
Target:
Glucagon Receptor

References

Decara JM, et al. Discovery of V-0219: A Small-Molecule Positive Allosteric Modulator of the Glucagon-Like Peptide-1 Receptor toward Oral Treatment for "Diabesity". J Med Chem. 2022 Apr 14;65(7):5449-5461.