TargetMol

Valorphin

Product Code:
 
TAR-T7306
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7306-2mg2mg£128.00
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TAR-T7306-5mg5mg£153.00
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TAR-T7306-10mg10mg£194.00
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TAR-T7306-25mg25mg£318.00
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TAR-T7306-50mg50mg£443.00
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Quantity:
TAR-T7306-100mg100mg£629.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
Valorphin has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 of 14 nM.
CAS:
144313-54-2
Formula:
C44H61N9O11
Molecular Weight:
892.024
Pathway:
GPCR/G Protein; Neuroscience; Endocrinology/Hormones
Purity:
0.98
SMILES:
CC(C)[C@H](N)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@@H]([C@@H](C)O)C(=O)N[C@@H](CCC(N)=O)C(O)=O
Target:
Opioid Receptor

References

Blishchenko E Y , Sazonova O V , Kalinina O A , et al. Antitumor effect of valorphin in vitro and in vivo: Combined action with cytostatic drugs[J]. Cancer Biology & Therapy, 2005, 4(1):125-131. Eyu B , Mernenko O A , Mirkina I I , et al. Tumor Cell Cytolysis Mediated by Valorphin, an Opioid-Like Fragment of Hemoglobin ?-Chain[J]. Peptides, 1997, 18(1):79-85.