TargetMol

Nelotanserin

Product Code:
 
TAR-T7350
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7350-1mg1mg£98.00
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TAR-T7350-2mg2mg£109.00
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TAR-T7350-1mL1 mL * 10 mM (in DMSO)£132.00
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TAR-T7350-5mg5mg£135.00
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TAR-T7350-10mg10mg£168.00
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TAR-T7350-25mg25mg£230.00
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TAR-T7350-50mg50mg£367.00
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TAR-T7350-100mg100mg£511.00
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TAR-T7350-500mg500mg£1,026.00
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Further Information

Bioactivity:
Nelotanserin is a potent 5-HT2A inverse agonist(IC50 : 1.7 nM), a moderately potent 5-HT2C partial inverse agonist t(IC50 :79 nM )and a weak 5-HT2B inverse agonistt(IC50 : 791 nM).
CAS:
839713-36-9
Formula:
C18H15BrF2N4O2
Molecular Weight:
437.245
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9842
SMILES:
COc1ccc(NC(=O)Nc2ccc(F)cc2F)cc1-c1c(Br)cnn1C
Target:
5-HT Receptor

References

Monti J M . Serotonin control of sleep-wake behavior[J]. Sleep Medicine Reviews, 2011, 15(4):0-281. Al-Shamma H A , Anderson C , Chuang E , et al. Nelotanserin, a Novel Selective Human 5-Hydroxytryptamine2A Inverse Agonist for the Treatment of Insomnia[J]. Journal of Pharmacology and Experimental Therapeutics, 2010, 332(1):281-290.