TargetMol

NPS2390

Product Code:
 
TAR-T8457
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8457-2mg2mg£100.00
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TAR-T8457-5mg5mg£118.00
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TAR-T8457-1mL1 mL * 10 mM (in DMSO)£140.00
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TAR-T8457-10mg10mg£148.00
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TAR-T8457-25mg25mg£222.00
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TAR-T8457-50mg50mg£334.00
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TAR-T8457-100mg100mg£503.00
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TAR-T8457-200mg200mg£666.00
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This product comes from: United States.
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Further Information

Bioactivity:
NPS2390 is a first generation quinoxaline derivative that acts as a noncompetitive antagonist of mGluR1 and mGluR5 (IC50 of 5.2 and 82 nM, respectively)
CAS:
226878-01-9
Formula:
C19H21N3O
Molecular Weight:
307.397
Pathway:
Neuroscience
Purity:
0.9924
SMILES:
O=C(NC12CC3CC(CC(C3)C1)C2)c1cnc2ccccc2n1
Target:
GluR

References

Peng X , Wei C , Li H Z , et al. NPS2390, a Selective Calcium-sensing Receptor Antagonist Controls the Phenotypic Modulation of Hypoxic Human Pulmonary Arterial Smooth Muscle Cells by Regulating Autophagy[J]. Journal of Translational Internal Medicine, 2019, 7(2):59-68.