TargetMol

DMU2139

Product Code:
 
TAR-T8728
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8728-1mg1mg£106.00
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TAR-T8728-2mg2mg£120.00
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TAR-T8728-5mg5mg£143.00
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TAR-T8728-1mL1 mL * 10 mM (in DMSO)£149.00
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TAR-T8728-10mg10mg£177.00
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TAR-T8728-25mg25mg£262.00
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TAR-T8728-50mg50mg£360.00
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TAR-T8728-100mg100mg£504.00
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This product comes from: United States.
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Further Information

Bioactivity:
DMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and 795 nM, respectively).
CAS:
104890-70-2
Formula:
C19H15NO2
Molecular Weight:
289.334
Pathway:
Metabolism
Purity:
0.9887
SMILES:
COc1ccc2cc(ccc2c1)C(=O)C=Cc1cccnc1
Target:
P45

References

Horley N J , Beresford K J M , Chawla T , et al. Discovery and characterization of novel CYP1B1 inhibitors based on heterocyclic chalcones: Overcoming cisplatin resistance in CYP1B1-overexpressing lines[J]. European Journal of Medicinal Chemistry, 2017, 129:159-174.