TargetMol

MM-102 TFA

Product Code:
 
TAR-T8768
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T8768-1mg1mg£97.00
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TAR-T8768-2mg2mg£108.00
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TAR-T8768-5mg5mg£156.00
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TAR-T8768-1mL1 mL * 10 mM (in DMSO)£193.00
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TAR-T8768-10mg10mg£213.00
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TAR-T8768-25mg25mg£310.00
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TAR-T8768-50mg50mg£426.00
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TAR-T8768-100mg100mg£595.00
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Further Information

Bioactivity:
MM-102 TFA is a potent WDR5/MLL interaction inhibitor, achieves IC50 = 2.4 nM. MM-102 compound prevents the interaction between mixed lineage leukemia 1 (MLL1) and WD Trp-Asp repeat domain 5 (WDR5) and results in the inhibition of MLL1 H3K4 histone methyltransferase (HMT) activity. Down-Regulation of H3K4me3 by MM-102 Facilitates Epigenetic Reprogramming of Porcine Somatic Cell Nuclear Transfer Embry
CAS:
1883545-52-5
Formula:
C37H50F5N7O6
Molecular Weight:
783.842
Pathway:
Chromatin/Epigenetic
Purity:
0.994
SMILES:
OC(=O)C(F)(F)F.CCC(CC)(NC(=O)C(C)C)C(=O)N[C@@H](CCCNC(N)=N)C(=O)NC1(CCCC1)C(=O)NC(c1ccc(F)cc1)c1ccc(F)cc1
Target:
Histone Methyltransferase

References

Karatas H, et al. J Am Chem Soc. 2013, 135(2), 669-682.