TargetMol

Venadaparib

Product Code:
 
TAR-T9430
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T9430-1mg1mg£103.00
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TAR-T9430-2mg2mg£116.00
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TAR-T9430-1mL1 mL * 10 mM (in DMSO)£148.00
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TAR-T9430-5mg5mg£148.00
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TAR-T9430-10mg10mg£189.00
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TAR-T9430-25mg25mg£309.00
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TAR-T9430-50mg50mg£462.00
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TAR-T9430-100mg100mg£646.00
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This product comes from: United States.
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Further Information

Bioactivity:
Venadaparib (IDX-1197) is a potent, selective and orally active PARP inhibitor with IC50s of 1.4 nM and 1.0 nM for PARP1 and PARP2, respectively. Venadaparib is insensitive to PARP-5. Venadaparib prevents the repair of DNA single-strand breaks (SSBs) and can be used in solid tumor research.
CAS:
1681017-83-3
Formula:
C23H23FN4O2
Molecular Weight:
406.461
Pathway:
DNA Damage/DNA Repair; Chromatin/Epigenetic
Purity:
0.9847
SMILES:
Fc1ccc(Cc2n[nH]c(=O)c3ccccc23)cc1C(=O)N1CC(CNC2CC2)C1
Target:
PARP

References

Cheng-Chang Chen, et al. A Small Molecule Restores Function to TRPML1 Mutant Isoforms Responsible for Mucolipidosis Type IV. Nat Commun. 2014 Aug 14;5:4681.