TargetMol

PF-06869206

Product Code:
 
TAR-TQ0011
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-TQ0011-2mg2mg£98.00
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TAR-TQ0011-1mL1 mL * 10 mM (in DMSO)£107.00
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TAR-TQ0011-5mg5mg£115.00
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TAR-TQ0011-10mg10mg£148.00
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TAR-TQ0011-25mg25mg£242.00
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TAR-TQ0011-50mg50mg£367.00
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Quantity:
TAR-TQ0011-100mg100mg£511.00
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Further Information

Bioactivity:
PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).
CAS:
2227425-05-8
Formula:
C15H14ClF3N4O2
Molecular Weight:
374.75
Pathway:
Membrane transporter/Ion channel
Purity:
1
SMILES:
Cc1[nH]c2c(N3CCO[C@H](CO)C3)c(C#N)c(nc2c1Cl)C(F)(F)F
Target:
Sodium Channel

References

Filipski KJ, et al. Discovery of Orally Bioavailable Selective Inhibitors of the Sodium-Phosphate Cotransporter NaPi2a (SLC34A1). ACS Med Chem Lett. 2018 Apr 12;9(5):440-445.