TargetMol

ABT-546

Product Code:
 
TAR-T10225
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10225-5mg5mg£850.00
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TAR-T10225-50mg50mg£1,661.00
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Quantity:
TAR-T10225-100mg100mg£2,079.00
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This product comes from: United States.
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Further Information

Bioactivity:
ABT-546 (A-216546) is a potent, highly selective, and active endothelin ETA receptor antagonist with a Ki of 0.46 nM for [125I]endothelin-1 binding to cloned human endothelin ETA.
CAS:
212481-66-8
Formula:
C30H48N2O6
Molecular Weight:
532.722
Purity:
0.98
SMILES:
CCCCN(CCCC)C(=O)CN1C[C@@H]([C@H]([C@@H]1CC(C)(C)CCC)C(O)=O)c1cc2OCOc2c(OC)c1

References

1. u-Wong JR, et al. Pharmacology of A-216546: a highly selective antagonist for endothelin ET(A) receptor. Eur J Pharmacol. 1999 Feb 5;366(2-3):189-201.