TargetMol

AR-A 2

Product Code:
 
TAR-T10360
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10360-5mg5mg£930.00
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TAR-T10360-50mg50mg£1,821.00
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Quantity:
TAR-T10360-100mg100mg£2,319.00
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Further Information

Bioactivity:
AR-A 2 is a selective 5-HT1B receptor antagonist, with a high affinity to guinea pig cortex 5HT1B/1D and recombinant guinea pig 5-HT1B receptors (Ki: 0.24 and 0.47 nM) and with 10-fold lower affinity to guinea pig 5-HT1D receptor (Ki: 5 nM).
CAS:
220051-79-6
Formula:
C27H36N4O2
Molecular Weight:
448.611
Purity:
0.98
SMILES:
CN1CCN(CC1)c1ccc(C)c2CC[C@H](Cc12)NC(=O)c1ccc(cc1)N1CCOCC1

References

1. Ahlgren C, et al. In vitro characterization of AR-A000002, a novel 5-hydroxytryptamine(1B) autoreceptor antagonist. Eur J Pharmacol. 2004 Sep 19;499(1-2):67-75.