TargetMol

AR453588 hydrochloride

Product Code:
 
TAR-T10362L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10362L-5mg5mg£1,091.00
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TAR-T10362L-50mg50mg£2,143.00
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Quantity:
TAR-T10362L-100mg100mg£2,801.00
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This product comes from: United States.
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Further Information

Bioactivity:
AR453588 hydrochloride is an orally bioavailable anti-diabetic glucokinase activator (EC50: 42 nM) with anti-hyperglycemic activity.
CAS:
1065606-97-4
Formula:
C25H26ClN7O2S2
Molecular Weight:
556.1
Purity:
0.98
SMILES:
Cl.CC(=O)N1CCC(CC1)c1nsc(Nc2ncc(Sc3ccccn3)cc2Oc2cccnc2C)n1

References

1. Hinklin RJ, et al. Discovery and preclinical development of AR453588 as an anti-diabetic glucokinase activator. Bioorg Med Chem. 2020 Jan 1;28(1):115232.