TargetMol

AVE5688

Product Code:
 
TAR-T10421
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10421-1mg1mg£449.00
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TAR-T10421-5mg5mg£670.00
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TAR-T10421-1mL1 mL * 10 mM (in DMSO)£852.00
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TAR-T10421-10mg10mg£1,026.00
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TAR-T10421-25mg25mg£1,492.00
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TAR-T10421-50mg50mg£1,990.00
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Quantity:
TAR-T10421-100mg100mg£2,657.00
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Further Information

Bioactivity:
AVE5688 is an inhibitor of glycogen phosphorylase (GP, IC50s: 430 nM and 915 nM; Kds: 170 nM and 530 nM for rmGPb and rmGPa). It can be used for the research of type 2 diabetes.
CAS:
613260-13-2
Formula:
C16H8ClF5N2O5
Molecular Weight:
438.69
Pathway:
Metabolism
Purity:
0.98
SMILES:
OC(=O)c1ccc(NC(=O)NC(=O)c2cc(F)c(F)cc2Cl)c(OC(F)(F)F)c1
Target:
Phosphorylase

References

1. Anderka O, et al. Thermodynamic characterization of allosteric glycogen phosphorylase inhibitors. Biochemistry. 2008 Apr 22;47(16):4683-91.