TargetMol

BR102375

Product Code:
 
TAR-T10596
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1

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CodeSizePrice
TAR-T10596-5mg5mg£850.00
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Quantity:
TAR-T10596-50mg50mg£1,661.00
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Quantity:
TAR-T10596-100mg100mg£2,079.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
BR102375 is a non-TZD PPAR γ full agonist (EC50: 0.28 μM) for the treatment of type 2 diabetes.
CAS:
2366255-59-4
Formula:
C31H34N6O4
Molecular Weight:
554.651
Purity:
0.98
SMILES:
CCCCc1nc(C)c(Cc2nc(no2)C(C)(C)C)c(=O)n1Cc1ccc(cc1)-c1ccccc1-c1noc(=O)[nH]1

References

1. Choung W, et al. Discovery of BR102375, a new class of non-TZD PPAR? full agonist for the treatment of type 2 diabetes. Bioorg Med Chem Lett. 2019 Jun 19. pii: S0960-894X(19)30407-X.