TargetMol

CARM1-IN-1

Product Code:
 
TAR-T10682L
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10682L-1mg1mg£104.00
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TAR-T10682L-5mg5mg£144.00
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TAR-T10682L-1mL1 mL * 10 mM (in DMSO)£160.00
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TAR-T10682L-10mg10mg£201.00
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TAR-T10682L-25mg25mg£332.00
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TAR-T10682L-50mg50mg£511.00
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Quantity:
TAR-T10682L-100mg100mg£704.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
CARM1-IN-1 is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows weak activity against PRMT1 and SET7 with IC50 > 600 μM.
CAS:
1020399-49-8
Formula:
C26H21Br2NO3
Molecular Weight:
555.26
Pathway:
Chromatin/Epigenetic
Purity:
0.9735
SMILES:
O=C1C(=CC2=CC=C(O)C(Br)=C2)CN(CC=3C=CC=CC3)CC1=CC4=CC=C(O)C(Br)=C4
Target:
Histone Methyltransferase

References

1. Cheng D, et al. Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity. J Med Chem. 2011 Jul 14;54(13):4928-32.