TargetMol

CB1 inverse agonist 1

Product Code:
 
TAR-T10694
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10694-1mg1mg£227.00
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TAR-T10694-5mg5mg£430.00
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TAR-T10694-1mL1 mL * 10 mM (in DMSO)£510.00
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TAR-T10694-10mg10mg£600.00
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TAR-T10694-25mg25mg£863.00
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TAR-T10694-50mg50mg£1,179.00
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TAR-T10694-100mg100mg£1,589.00
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TAR-T10694-500mg500mg£3,115.00
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Further Information

Bioactivity:
CB1 inverse agonist 1 is an orally active, and specific inverse agonist of the CB1 receptor (IC50s: 7.5 nM and 4100 nM for CB1 and CB2 receptors) with anorexigenic effects.
CAS:
852315-00-5
Formula:
C25H18Cl3N3O3
Molecular Weight:
514.79
Pathway:
GPCR/G Protein
Purity:
0.98
SMILES:
CC(=O)Nc1c(C(C)=O)c(=O)n(C)c2nc(-c3ccc(Cl)cc3Cl)c(cc12)-c1ccc(Cl)cc1
Target:
Cannabinoid Receptor

References

1. Debenham JS, et al. Synthesis of functionalized 1,8-naphthyridinones and their evaluation as novel, orally active CB1 receptor inverse agonists.Bioorg Med Chem Lett. 2006 Feb;16(3):681-5.