TargetMol

CBP/p300-IN-2

Product Code:
 
TAR-T10702
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10702-5mg5mg£1,572.00
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TAR-T10702-50mg50mg£3,107.00
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Quantity:
TAR-T10702-100mg100mg£4,247.00
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This product comes from: United States.
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  • Further Information
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Further Information

Bioactivity:
CBP/EP300-IN-2 is an inhibitor of CBP/EP300 (IC50s: 1.07 nM and 5.96 nM for CBP/HTRF and Myc) extracted from patent WO2017205538A1 (example 25).
CAS:
2158265-96-2
Formula:
C27H29F2N7O2
Molecular Weight:
521.573
Pathway:
Chromatin/Epigenetic; Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
CNC(=O)N1CCc2c(C1)c(nn2C1CCOCC1)-c1cncc2cc(-c3cnn(C)c3)c(cc12)C(F)F
Target:
Epigenetic Reader Domain; c-Myc

References

1. Patrick Cyr, et al. Pyrazolopyridine derivatives for the treatment of cancer