TargetMol

CPUY074020

Product Code:
 
TAR-T10882
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10882-1mg1mg£227.00
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TAR-T10882-5mg5mg£431.00
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TAR-T10882-1mL1 mL * 10 mM (in DMSO)£468.00
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TAR-T10882-10mg10mg£600.00
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TAR-T10882-25mg25mg£863.00
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TAR-T10882-50mg50mg£1,187.00
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Quantity:
TAR-T10882-100mg100mg£1,581.00
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TAR-T10882-500mg500mg£3,107.00
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This product comes from: United States.
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Further Information

Bioactivity:
CPUY074020 is a potent and orally bioavailable inhibitor of histone methyltransferase G9a (IC50: 2.18 μM) with anti-proliferative activity.
CAS:
902279-44-1
Formula:
C25H28N4O2
Molecular Weight:
416.525
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
O=C1c2ccccc2-c2onc3c(cc(NCCN4CCCC4)c1c23)N1CCCCC1
Target:
Histone Methyltransferase

References

1. Chen WL, et al. Discovery, design and synthesis of 6H-anthra[1,9-cd]isoxazol-6-one scaffold as G9a inhibitor through a combination of shape-based virtual screening and structure-based molecular. Bioorg Med Chem. 2016 Nov 15;24(22):6102-6108.