TargetMol

CS-003 Free base

Product Code:
 
TAR-T10892
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10892-5mg5mg£1,412.00
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TAR-T10892-50mg50mg£2,785.00
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Quantity:
TAR-T10892-100mg100mg£3,765.00
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Further Information

Bioactivity:
CS-003 free base (CS-003) is a triple tachykinin receptor antagonist with high affinity for human (neurokinin) NK1, NK2 and NK3 receptors, with Ki values of 2.3 nM and 0.54 nM, respectively And 0.74 nM. CS-003 free base (CS-003) has therapeutic effects on neurokinin-related respiratory diseases.
CAS:
191672-52-3
Formula:
C34H38Cl2N2O6S
Molecular Weight:
673.65
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.98
SMILES:
COc1cc(cc(OC)c1OC)C(=O)N1CCOC(CCN2CCC3(CC2)c2ccccc2CS3=O)(C1)c1ccc(Cl)c(Cl)c1
Target:
Neurokinin receptor

References

1. Tsuchida H, et al. Novel triple neurokinin receptor antagonist CS-003 strongly inhibits neurokinin related responses. Eur J Pharmacol. 2008 May 31;586(1-3):306-12.