TargetMol

DSP-1053

Product Code:
 
TAR-T11107
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11107-5mg5mg£463.00
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Quantity:
TAR-T11107-50mg50mg£2,062.00
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Quantity:
TAR-T11107-100mg100mg£3,267.00
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This product comes from: United States.
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Further Information

Bioactivity:
Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.
CAS:
1176326-76-3
Formula:
C26H32BrNO4
Molecular Weight:
502.449
Purity:
0.98
SMILES:
COCCOc1cc(CC2CCN(CCc3ccc4OCCC(=O)c4c3)CC2)ccc1Br

References

1. Yoshinaga H, et al. Discovery of DSP-1053, a novel benzylpiperidine derivative with potent serotonin transporter inhibitory activity and partial 5-HT1A receptor agonistic activity. Bioorg Med Chem. 2018 May 1;26(8):1614-1627.