TargetMol

Endomorphin 2 TFA

Product Code:
 
TAR-T11198
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11198-5mg5mg£124.00
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TAR-T11198-10mg10mg£164.00
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TAR-T11198-25mg25mg£271.00
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Further Information

Bioactivity:
Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM. a high affinity, highly selective agonist of the μ-opioid receptor,
CAS:
1276124-00-5
Formula:
C34H38F3N5O7
Molecular Weight:
685.701
Pathway:
Endocrinology/Hormones; Neuroscience; GPCR/G Protein
Purity:
0.98
SMILES:
OC(=O)C(F)(F)F.N[C@@H](Cc1ccc(O)cc1)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Target:
Opioid Receptor

References

1. Goldberg IE, et al. Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse brain. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.