TargetMol

GPR120 Agonist 1

Product Code:
 
TAR-T11452
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11452-5mg5mg£1,010.00
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TAR-T11452-50mg50mg£1,982.00
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Quantity:
TAR-T11452-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GPR120 (the calcium flux assay), respectively.
CAS:
1628448-77-0
Formula:
C20H12ClF6NO3S
Molecular Weight:
495.82
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.98
SMILES:
OC(=O)CCc1cc(F)c(OCc2c(nsc2C(F)(F)F)-c2ccc(Cl)cc2F)c(F)c1
Target:
GPR

References

1. Zhang X, et al. Discovery of an Isothiazole-Based Phenylpropanoic Acid GPR120 Agonist as a Development Candidate for Type 2 Diabetes. ACS Med Chem Lett. 2017 Jul 27;8(9):947-952.